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Stereocontrolled synthesis of the cis‐hydroxydecalin system: Towards biologically active 19‐nor‐clerodanes
Mirzayans, P. M.; Pouwer, R. H.; Williams, C. M.; Bernhardt, P. V.; Eur. J. Org. Chem., 2012, 2012(8), 1633-1638
Diastereoselective 1,3-dipolar cycloaddition of pyrylium ylides with chiral enamides
Tchabanenko, K.; Sloan, C.; Bunetel, Y.; Mullen, P.; Org. Bioorg. Chem., 2012, 10, 4215-4219
Using continuous processes to increase production
Anderson, N. G.; Org. Process Res. Dev., 2012, 16(5), 852-869
Synthesis of a new family of acyclic nucleoside phosphonates, analogues of TPases transition states
Dayde, B.; Benzaria, S.; Pierra, C.; Gosselin, G.; Surleraux, D.; Volle, J.; Pirat, J.; Virieux, D.; Org. Biomol. Chem, 2012, 10, 3448-3454
Synthesis of amines from alcohols in a nonepimerizing one-pot sequence – Synthesis of bioactive compounds: Cinacalcet and dexoxadrol
Guerin, C.; Bellosta, V.; Guillamot, G.; Cossy, J.; Eur. J. Org. Chem., 2012, 15, 2990-3000
Continuous flow synthesis. A pharma perspective
Malet-Sanz, L.; Susanne, F.; J. Med. Chem., 2012, 55(9), 4062-4098
Process development of a potent glucosylceramide synthase inhibitor
Cooper, C. G. F.; Lee, E. R.; Silva, R. A.; Bourque, A. J.; Clark, S.; Katti, S.; Nivorozkhin, V.; Org. Process Res. Dev., 2012, 16(5), 1090-1097
Reductive amination by continuous-flow hydrogenation: direct and scalable synthesis of a benzylpiperazine
Liu, J.; Fitzgerald, A. E.; Mani, N. S.; Synthesis, 2012, 44(15), 2469-2473
Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist
Xiong, H.; Wu, Y.; Lehr, S. G.; Blackwell, W.; Steelman, G.; Hulsizer, J.; Urbanek, R. A.; Tetrahedron Letters, 2012, 53(44), 5833-5836