Synthesis, SAR, and pharmacological characterization of brain penetrant P2X7 receptor antagonists

Savall, B. M.; Wu, D.; Angelis, M. D.; Carruhters, N. I.; Ao, H.; Wang, Q.; Lord, B.; Bharrachrya, A.; Letavic, M. A.; ACS Med. Chem. Lett., 2015, 6, 671-676

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