Total synthesis and biological evaluation of tubulysin analogues

Colombo, R.; Wang, Z.; Han, J.; Balachandran, R.; Daghestani, H. N.; Camarco, D. P.; Vogt, A.; Day, B. W.; Mendel, D.; Wipf, P.; J. Org. Chem., 2016, 81(21), 10302-10320

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