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Synthesis of amines from alcohols in a nonepimerizing one-pot sequence – Synthesis of bioactive compounds: Cinacalcet and dexoxadrol
Guerin, C.; Bellosta, V.; Guillamot, G.; Cossy, J.; Eur. J. Org. Chem., 2012, 15, 2990-3000
Continuous flow synthesis. A pharma perspective
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Process development of a potent glucosylceramide synthase inhibitor
Cooper, C. G. F.; Lee, E. R.; Silva, R. A.; Bourque, A. J.; Clark, S.; Katti, S.; Nivorozkhin, V.; Org. Process Res. Dev., 2012, 16(5), 1090-1097
Reductive amination by continuous-flow hydrogenation: direct and scalable synthesis of a benzylpiperazine
Liu, J.; Fitzgerald, A. E.; Mani, N. S.; Synthesis, 2012, 44(15), 2469-2473
Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist
Xiong, H.; Wu, Y.; Lehr, S. G.; Blackwell, W.; Steelman, G.; Hulsizer, J.; Urbanek, R. A.; Tetrahedron Letters, 2012, 53(44), 5833-5836
Synthesis of a biphenyl library for studies of hydrogen bonding in the solid state
Baltus, C. B.; Press, N. J.; Antonijevic, M. D.; Tizzard, G. J.; Coles, S. J.; Spencer, J.; Tetrahedron, 2012, 68(45), 9272-9277
Synthesis and arylation of unprotected sulfonimidamides
Maldonado; M. F.; Sehgelmeble, F.; Bjarnemark, F.; Svensson, M.; Ahman, F.; Arvidsson, P. I.; Tetrahedron, 2012, 68, 7456-7462
A method to identify best available technologies (BAT) for hydrogenation reactors in the pharmaceutical industry
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Modeling, synthesis and biological evaluation of potential retinoid X receptor‐selective agonists: Novel halogenated analogues of 4‐[1‐(3,5,5,8,8‐pentamethyl‐5,6,7,8‐tetrahydro‐2‐naphthyl)ethynyl]benzoic acid (Bexarotene)
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