Brasholz, M.; Macdonald, J. M.; Saubern, S.; Ryan, J. H.; Holmes, A. B.; Chem. Eur. J., 2010, 16(37), 11471-11480
Lipase-catalyzed kinetic resolution of 2-methylene-substituted cycloalkanols in batch and continuous-flow modes
Tomin, A.; Hornyanszky, G.; Kupai, K.; Dorko, Zs.; Urge, L.; Darvas, F.; Poppe, L.; Process Biochemistry, 2010, 45(6), 859-865
Straightforward hetero Diels-Alder reactions of nitroso dienophiles by microreactor technology
Monbaliu, J-C. M. R.; Cukalovic, A.; Marchand-Brynaert, J.; Stevens, C. V.; Tetrahedron Letters, 2010, 51, 5830-5833
Reversal of the ee in enantioselective hydrogenation of activated ketones in continuous-flow fixed-bed reactor system
Cserenyi, Sz.; Szollosi, Gy.; Szori, K.; Fulop, F.; Bartok, M.; Catalysis Communications, 2010, 12, 14-19
Synthesis of a tetrasaccharide related to the triterpenoid saponin Bellisoside isolated from Bellis perennis (compositae)
Mandal, S.; Sharma, N.; Mukhopadhyay, B.; Tetrahedron: Asymmetry, 2010, 21, 2172-2176
Novel spirotetracyclic zwitterionic dual H1/5-HT2A receptor antagonists for the treatment of sleep disorders
Gianotti, M.; Botta, M.; Brough, S.; Carletti, R.; Castiglioni, E.; Corti, C.; Dal-Cin, M.; Fratte, S. D.; Korajec, D.; Lovric, M.; Merlo, G.; Mesic, M.; Pavone, F.; Piccoli, L.; Rast, S.; Roscic, M.; Sava, A.; Smehil, M.; Stasi, L.; Togninelli, A.; Wigglesworth, M. J.; J. Med. Chem., 2010, 53, 7778-7795
Aminopyrazine inhibitors binding to an unusual inactive conformation of the mitotic kinase Nek2: SAR and structural characterization
Whelligan, D. K.; Solanki, S.; Taylor, D.; Thomson, D. W.; Cheung, K. J.; Boxall, K.; Mas-Droux, C.; Barillari, C.; Burns, S.; Grummitt, C. G.; Collins, I.; van Montfort, E. L. M.; Aherne, G. W.; Bayliss, R.; Hoelder, S.; J. Med. Chem., 2010, 53, 7682-7698
Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity
Borcard, F.; Baud, M.; Bello, C.; Dal Bello, G.; Grossi, F.; Pronzato, P.; Cea, M.; Nencioni, A.; Vogel, P.; Bioorg. Med. Chem. Lett., 2010, 20(17), 5353-5356
Synthesis of functionalized 3-hydroxypiperidines
Wijdeven, M. A.; van Delft, F. L.; Rutjes, F. P. J. T.; Tetrahedron, 2010, 66, 5623-5636