De novo design of a picomolar nonbasic 5-HT1B receptor antagonist

Nugiel, D. A.; Krumrine, J. R.; Hill, D. C.; Damewood, J. R.; Bernstein, P. R.; Sobotka-Briner, C. D.; Liu, J. W.; Zacco, A.; Pierson, M. E.; J. Med. Chem., 2010, 53, 1876-1880

Link to article