Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and cocrystal structure

Milite, C.; Feoli, A.; Horton, J. R.; Rescigno, D.; Cipriano, A.; Pisapia, V.; Viviano, M.; Pepe, G.; Amendola, G.; Novellino, E.; Cosconati, S.; Cheng, X.; Castellano, S.; Sbardella, G.; J. Med. Chem., 2019, 62(5), 2666-2689

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