3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis

Ferrins, L.; Rahmani, R.; Sykes, M. L.; Jones, A. J.; Avery, V. M.; Teston, E.; Almohaywi, B.; Yin, J.; Smith, J.; Hyland, C.; White, K. L.; Ryan, E.; Campbell, M.; Charman, S. A.; Kaiser, M.; Baell, J. B.; Eur. J. Med. Chem., 2013, 66, 450-465

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Synthesis and biological evaluation of 2,3-diarylimidazo[1,2-a]pyridines as antileishmanial agents

Marhadour, S.; Marchand, P.; Pagniez, F.; Bazin, M. A.; Picot, C.; Lozach, O.; Ruchaud, S.; Antoine, M.; Meijer, L.; Rachidi, N.; Le Pape, P.; Eur. J. Med. Chem., 2012, 58, 543-556

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A remote-controlled adaptive medchem lab: an innovative approach to enable drug discovery in the 21st Century

Godfrey, A. G.; Masquelin, T.; Hemmerle, H.; Drug Discovery Today, 2013, 18(17-18), 795-802

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Design of a highly selective and potent class of non-planar estrogen receptor ß agonists

Sunden, H.; Ma, J. N.; Hansen, L. K.; Gustavsson, A. L.; Burstein, E. S.; Olsson, R.; ChemMedChem, 2013, 8(8), 1283-1294

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Site‐selective deuterated‐alkene synthesis with palladium on boron nitride

Yabe, Y.; Sawama, Y.; Monguchi, Y.; Sajiki, H.; Chem. Eur. J., 2013, 19, 484-488

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Multistep continuous‐flow synthesis in medicinal chemistry: Discovery and preliminary structure-activity relationships of CCR8 ligands

Petersen, T. P.; Mirsharghi, S.; Rummel, P. C.; Thiele, S.; Rosenkilde, M. M.; Ritzen, A.; Ulven, T.; Chem. Eur. J., 2013, 19(28), 9343-9350

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Total synthesis, stereochemical assignment, and biological activity of chamuvarinin and structural analogues

Florence, G. J.; Morris, J. C.; Murray, R. G.; Vanga, R. R.; Osler, J. D.; Smith, T. K.; Chem. Eur. J., 2013, 19, 8309-8320

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Reversible and efficient inhibition of UDP‐galactopyranose mutase by electrophilic, constrained and unsaturated UDP‐galactitol analogues

Ansiaux, C.; N’Go, I.; Vincent, S. P.; Chem. Eur. J., 2012, 18(46), 14860-14866

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Rapid microfluidic flow hydrogenation for reduction or deprotection of 18F-labeled compounds

Liang, S. H.; Collier, T. L.; Rotstein, B. H.; Lewis, R.; Steck, M.; Vasdev, N.; Chem. Commun., 2013, 49(78), 8755-8757

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Single operation stereoselective synthesis of Aerangis lactones: Combining continuous flow hydrogenation and biocatalysts in a chemoenzymatic sequence

Fink, M. J.; Schon, M.; Rudroff, F.; Schnurch, M.; Mihovilovic, M. D.; ChemCatChem, 2013, 5, 724-727

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